Compile Data Set for Download or QSAR
maximum 50k data
Found 17 of ki data for polymerid = 50001945,50006714
TargetPyruvate kinase PKLR(Homo sapiens (Human))
Universit£ di Pisa

Curated by ChEMBL
LigandPNGBDBM50336799(5,5',5''-[1,3,6-naphthalenetriyltris(sulfonylimino...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367052(CHEMBL605425)
Affinity DataKi:  1.60E+6nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-L)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367051(CHEMBL606059)
Affinity DataKi:  2.20E+6nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-K)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028624(CHEMBL3142978 | [6-(6-amino-9H-purin-9-yl)-2-methy...)
Affinity DataKi:  2.20E+6nMAssay Description:Inhibition of rat liver pyruvate kinase (PK-L) at 3.6 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367051(CHEMBL606059)
Affinity DataKi:  2.20E+6nMAssay Description:Inhibition of rat muscle pyruvate kinase (PK-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367051(CHEMBL606059)
Affinity DataKi:  2.90E+6nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-K)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367052(CHEMBL605425)
Affinity DataKi:  3.80E+6nMAssay Description:Inhibitory constant for inhibition of pyruvate kinase obtained from rat liver (PK-L) was determined using ADP as competitive inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367054(CHEMBL606476)
Affinity DataKi:  3.90E+6nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-K) at 6.7 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028624(CHEMBL3142978 | [6-(6-amino-9H-purin-9-yl)-2-methy...)
Affinity DataKi:  4.60E+6nMAssay Description:Inhibition of rat liver pyruvate kinase (PK-L); (relative inhibitory potency)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367053(CHEMBL605428)
Affinity DataKi:  5.00E+6nMAssay Description:Inhibition of rat muscle pyruvate kinase (PK-M) at 6.7 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367050(CHEMBL606006)
Affinity DataKi:  5.40E+6nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-K)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028625(CHEMBL3142968 | [5-(6-amino-9H-purin-9-yl)-4-hydro...)
Affinity DataKi:  7.00E+6nMAssay Description:Inhibitory constant for inhibition of pyruvate kinase obtained from rat liver (PK-L) was determined using ADP as competitive inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367053(CHEMBL605428)
Affinity DataKi:  7.50E+6nMAssay Description:Inhibitory constant for inhibition of pyruvate kinase obtained from rat liver (PK-L) was determined using ADP as competitive inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367050(CHEMBL606006)
Affinity DataKi:  8.00E+6nMAssay Description:Michaelis-Menten constant for inhibition of rat kidney pyruvate kinase (PK-K)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367054(CHEMBL606476)
Affinity DataKi:  8.40E+6nMAssay Description:Inhibitory constant for inhibition of pyruvate kinase obtained from rat liver (PK-L) was determined using ADP as competitive inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367050(CHEMBL606006)
Affinity DataKi:  1.09E+7nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-K) at 6.7 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028625(CHEMBL3142968 | [5-(6-amino-9H-purin-9-yl)-4-hydro...)
Affinity DataKi:  3.20E+7nMAssay Description:Inhibition of rat kidney pyruvate kinase (PK-K)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed